Synthesis of 2?,3?-modified carbocyclic L -nucleoside analogues

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Autor/in:
Erscheinungsjahr:
2011
Medientyp:
Text
Schlagworte:
  • Nucleosides
  • Antiviral Agents
  • Carbocyclic nucleosides
  • Oligonucleotides
  • DNA
  • Nucleosides
  • Antiviral Agents
  • Carbocyclic nucleosides
  • Oligonucleotides
  • DNA
Beschreibung:
  • New divergent approaches to 2',3'-modified carbocyclic L-nucleoside analogues starting from enantiomerically pure (1R, 2S)- or (1S, 2R)-2-(benzyloxymethyl) cyclopent-3-enol are described. In the key step, stereochemically pure cyclopentanols were condensed with N3-protected thymine through a modified Mitsunobu protocol. Moreover, several routes to different cyclopentanol derivatives, to prepare carbocyclic L-2',3'-didehydro-2',3'-dideoxynucleosides (L-d4N), L-2',3' -dideoxynucleosides (L-ddN), and L-ribonucleosides are reported.
Lizenz:
  • info:eu-repo/semantics/restrictedAccess
Quellsystem:
Forschungsinformationssystem der UHH

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Quelldatensatz
oai:www.edit.fis.uni-hamburg.de:publications/0865f385-e289-406b-b67c-83a1e4eca078