Pd-Catalyzed Synthesis of γ-Keto Esters as Key Intermediates for the Synthesis of γ-Hydroxybutenolides

Link:
Autor/in:
Erscheinungsjahr:
2019
Medientyp:
Text
Schlagworte:
  • Boronic acids
  • Carbonylation
  • Catalysis
  • Cross-coupling
  • Vinyltosylates
Beschreibung:
  • We herein report a robust and safe palladium catalyzed domino‐carbonylation/Suzuki–Miyaura cross‐coupling reaction of vinyltosylates with arylboronic acids using Mo(CO)6 as CO‐source. The derived γ‐keto ester were subsequently cyclized under acidic conditions to obtain γ‐hydroxybutenolides, an important structural motif, which occurs in biologically active natural products.
Lizenz:
  • info:eu-repo/semantics/restrictedAccess
Quellsystem:
Forschungsinformationssystem der UHH

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Quelldatensatz
oai:www.edit.fis.uni-hamburg.de:publications/43257915-d215-4a2a-aabb-7af3642db1e1